先导化合物|Lead compound
先导化合物
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1-cyclopropyl-7-(3-((ethylamino)methyl)pyrrolidin-1-yl)-6,8-difluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
CAS号:99734-97-1
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3-((3-methylbenzyl)(3-phenoxybenzyl)amino)propanoic acid
CAS号:434910-94-8
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1-(3,4-dimethoxyphenyl)-3-(3-imidazol-1-ylpropyl)thiourea
CAS号:790663-33-1
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(5S,8S,14S,17S,20S)-14-((1H-indol-3-yl)methyl)-20-(((S)-1-amino-1-oxo-3-phenylpropan-2-yl)carbamoyl)-8,17-dibutyl-16-methyl-3,6,11,12,15,18-hexaoxo-5-(4-(sulfooxy)benzyl)-4,7,9,13,16,19-hexaazadocosan-22-oic-1,1,1,2,2-t5 acid
CAS号:125236-85-3
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Ethanesulfonic acid, 2-((2,4-dihydroxy-3,3-dimethyl-1-oxobutyl)amino)-, (R)- (9CI)
CAS号:2545-84-8
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2-Naphthoic acid, 4,4'-methylenebis(3-hydroxy-, compd. with 8-((4-(diethylamino)-1-methylbutyl)amino)-6-methoxyquinoline (11)
CAS号:635-05-2
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Benzoic acid, 2-hydroxy-6-methyl-, [(1S,2R,3R,4S,5S)-5-[(3-acetylphenyl)amino]-4-amino-3-[[(dimethylamino)carbonyl]amino]-1,2-dihydroxy-3-[(1S)-1-hydroxyethyl]-2-methylcyclopentyl]methyl ester
CAS号:23668-11-3
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N-(3-Methoxypropyl)-7-methyl-4-oxo-4,5-dihydro-[1,2,3]triazolo[1,5-a]quinoxaline-3-carboxamide
CAS号:1359627-33-0
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9-Octadecenoic acid, 2-((2-amino-1,6-dihydro-6-oxo-9H-purin-9-yl)methoxy)ethyl ester, (E)-
CAS号:151090-37-8
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Carbamic acid, ((1S)-2-(((5S)-5-(((4-aminophenyl)sulfonyl)(2-methylpropyl)amino)-6-hydroxyhexyl)amino)-1-(1H-indol-3-ylmethyl)-2-oxoethyl)-, methyl ester
CAS号:449806-40-0
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4,5-Bis(4-methoxyphenyl)-1,3-dihydroimidazol-2-one
CAS号:71727-40-7
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trans-4-[8-amino-1-(7-chloro-1H-indol-2-yl)imidazo[1,5-a]pyrazin-3-yl]-cyclohexanecarboxylic acid
CAS号:936889-68-8
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(S)-2-(dimethylamino)-3-(4-mercapto-1-methyl-1H-imidazol-5-yl)propanoic acid
CAS号:105496-34-2
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(S)-2-amino-3-(4-mercapto-1-methyl-1H-imidazol-5-yl)propanoic acid
CAS号:108418-13-9
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4-[6-Amino-7-[[(R)-1-(2,6-dichloro-3-fluorophenyl)ethyl]oxy]furo[3,2-c]pyridin-3-yl]-3,6-dihydro-2H-pyridine-1-carboxamide
CAS号:1175296-94-2
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5-Amino-N-(1,1-dimethylethyl)-2-(methylthio)-4-[3-[[2-(4-morpholinyl)acetyl]amino]phenyl]thieno[2,3-d]pyrimidine-6-carboxamide
CAS号:501444-88-8
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(4S,7S,10S,13R,16S)-7-((1H-imidazol-4-yl)methyl)-4-(2-aminobutanamido)-13-(4-aminobutyl)-10,16-dibenzyl-19-butyl-2-(methylsulfinyl)-5,8,11,14,17-pentaoxo-18-oxa-6,9,12,15-tetraazatetracosanoic acid
CAS号:132031-83-5
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(2S)-2,6-diamino-5-(phosphonooxy)hexanoic acid
CAS号:32163-95-4
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Pyrazine, 1-(3,4-dimethoxybenzoyl)-1,2,3,4-tetrahydro-4-(1,2,3,4-tetrahydro-2-oxo-6-quinolinyl)-
CAS号:211369-52-7
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6-[(2R,3S)-3-[[[(4-Chloro-2-methylphenyl)sulfonyl]amino]methyl]bicyclo[2.2.2]oct-2-yl]-5Z-hexenoic acid
CAS号:216158-34-8
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(Z)-2-((6-methyl-5-(2-(((phenyl(pyridin-3-yl)methylene)amino)oxy)ethyl)-7,8-dihydronaphthalen-1-yl)oxy)acetic acid
CAS号:176391-41-6
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Propan-2-yl N-(6-((N-((4-(1H-pyrazol-1-yl)phenyl)methyl)pyridine-3-sulfonamido)methyl)pyridin-2-yl)glycinate
CAS号:1187451-19-9
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3-Quinolinecarboxylic acid, 5-amino-7-(7-amino-5-azaspiro(2,4)hept-5-yl)-1-cyclopropyl-6-fluoro-1,4-dihydro-8-methyl-4-oxo-, (S)-
CAS号:167887-97-0
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(R)-1-(1-((S)-Tetrahydro-2H-pyran-3-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl)ethan-1-ol
CAS号:1315485-91-6
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O8 OGG1 Inhibitor
CAS号:350997-39-6
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(2S)-2-amino-5-((hydroxy(sulfamoyloxy)phosphoryl)amino)pentanoic acid
CAS号:65370-68-5
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(S)-2-amino-3-(2-((bis(2-chloroethyl)amino)methyl)phenyl)propanoic acid hydrochloride
CAS号:2185-98-0
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(S)-2-amino-3-(2-((bis(2-chloroethyl)amino)methyl)phenyl)propanoic acid
CAS号:3734-80-3
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5-(1,1-Dimethylheptyl)-2-(4-phenylcyclohexyl)-1,3-benzenediol
CAS号:468083-84-3
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1-methylimidazolidine-2,4-dione
CAS号:84210-26-4
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(S)-3-ethyl-9,10-dimethoxy-2-(((R)-1,2,3,4-tetrahydroisoquinolin-1-yl)methyl)-1,6,7,11b-tetrahydro-4H-pyrido[2,1-a]isoquinoline
CAS号:75041-32-6
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3(S)-[2-Chloro-5-(2,2-difluoro-ethyl)-8-fluoro-5H-dibenzo[b,e][1,4]diazepin-11-ylamino]-pyrrolidine-1-carboxylic acid isopropylamide
CAS号:1783816-74-9
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(2S)-2-[(2S)-2-amino-3-methylbutanamido]-3-(1H-indol-3-yl)propanoic acid
CAS号:24587-37-9
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8-[2-Methoxy-4-(4-methyl-piperazin-1-yl)-phenylamino]-4,5-dihydro-7,9,9b-triaza-cyclopenta[a]naphthalene-3-carboxylic acid (2,6-diethyl-phenyl)-amide
CAS号:1817791-73-3
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3,9-Dihydro-8-methoxy-9-methyl-2-(1-methylethyl)furo(2,3-b)quinolin-4(2H)-one
CAS号:52486-77-8
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N1,N4-bis(3-(1H-benzo[d]imidazol-2-yl)phenyl)terephthalamide
CAS号:500538-94-3
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2-Chloro-4',4''-di-2-imidazolin-2-yl-terephthalanilide
CAS号:70-09-7
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((S)-4-carboxy-4-(4-(((2,4-diaminopteridin-6-yl)methyl)(methyl)amino)benzamido)butanoyl)-L-glutamic acid
CAS号:41600-13-9
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(4-(((2,4-diaminopteridin-6-yl)methyl)(methyl)amino)-1-naphthoyl)-L-glutamic acid
CAS号:136242-96-1
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(4-(((2,4-diaminopteridin-6-yl)methyl)(methyl)amino)-3-methoxybenzoyl)-L-glutamic acid
CAS号:82144-26-1


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