先导化合物|Lead compound
先导化合物
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3-[6-[(4-Methylpiperazin-1-yl)methyl]-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl]phenol
CAS号:885616-78-4
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5,7-Dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-8-(1-methylpyrrolidin-2-yl)chromen-4-one
CAS号:76540-48-2
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N-(3,5-Dimethyl-phenyl)-3-(4-oxo-3,4,5,6,7,8-hexahydro-benzo[4,5]thieno[2,3-d]pyrimidin-2-yl)-propionamide
CAS号:1003736-23-9
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Phosphoric acid, mono(4-nitrophenyl) ester, compd. with 2-amino-2-ethyl-1,3-propanediol (12)
CAS号:62796-28-5
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4-氨基-3-苯基丁酸盐酸盐
CAS号:1078-21-3
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D-3,4-Dimethyl-2-phenyl-morpholine tartrate
CAS号:50-58-8
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Phosphonic acid, (3-amino-2-(4-chlorophenyl)propyl)-
CAS号:108351-35-5
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N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-pyrrolidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide
CAS号:900305-37-5
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4-[4-(4,6-Dimethyl-5-pyrimidinyl)-3-methylphenoxy]-1H-pyrazolo[4,3-c]pyridine
CAS号:1609258-91-4
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Isoquinoline, 1-(2-(3,4-dimethoxyphenyl)ethyl)-3,4-dihydro-6-methyl-, hydrochloride
CAS号:132928-46-2
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Ketohexokinase Inhibitor 1
CAS号:2102501-84-6
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2-[[trans-4-[2-Amino-6-(6-methoxy-3-pyridinyl)-4-methyl-7-oxopyrido[2,3-d]pyrimidin-8(7H)-yl]cyclohexyl]oxy]acetic acid
CAS号:1431626-44-6
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4-[5-(1-methylpyrazol-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]morpholine
CAS号:1527473-30-8
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2-((S)-1-(4-fluoro-2-((R)-1,1,1-trifluoropropan-2-yl)phenoxy)propan-2-yl)-7-(4-methyl-1H-imidazol-1-yl)-3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-dione
CAS号:1402002-76-9
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1-Methyl-6-(2-pyridinylmethoxy)-3-[4-(trifluoromethyl)-3-pyridinyl]-1H-pyrazolo[3,4-b]prazine
CAS号:1539296-46-2
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(R)-3-(4-((3,3-dimethylcyclobutyl)((6-(4-(trifluoromethyl)-1H-imidazol-1-yl)pyridin-3-yl)amino)methyl)benzamido)propanoic acid
CAS号:1407592-99-7
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6-[(2,5-Dimethoxyphenyl)thio]-3-(1-methyl-1H-pyrazol-4-yl)-1,2,4-triazolo[4,3-b]pyridazine
CAS号:1622291-81-9
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1-Methyl-3-(4-methyl-3-pyridinyl)-6-(2-pyridinylmethoxy)-1H-pyrazolo[3,4-b]pyrazine
CAS号:1539296-45-1
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2-(1H-Benzimidazol-1-ylmethyl)-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
CAS号:1434288-24-0
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(R)-6-(4-methyl-1,1-dioxido-1,2,6-thiadiazinan-2-yl)isoquinoline-1-carbonitrile
CAS号:1612755-71-1
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5-Methyl-3-[[(2R)-4-(2-thiazolylmethyl)-2-morpholinyl]methyl]-3H-1,2,3-triazolo[4,5-d]pyrimidin-7-amine hydrochloride
CAS号:1305116-67-9
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5-Methyl-3-[[(2R)-4 (2-thiazolylmethyl)-2-morpholinyl]methyl]-3H-1,2,3-triazolo[4,5-d]pyrimidin-7-amine
CAS号:1305116-69-1
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1-[(1S)-1-[2-[[[[3,5-Bis(trifluoromethyl)phenyl]methyl](2-methyl-2H-tetrazol-5-yl)amino]methyl]-4-(trifluoromethyl)phenyl]-2-methylpropyl]-4-piperidinecarboxylic acid
CAS号:949099-81-4
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1H-Pyrazolo(4,3-d)pyrimidine-3-carboxamide, 1-(2-ethoxyethyl)-5-(ethylmethylamino)-7-((4-methyl-2-pyridinyl)amino)-N-(methylsulfonyl)
CAS号:853003-48-2
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(2S,5S,8S,11S,14S,17S,20S,23S,26S)-20-((1H-indol-3-yl)methyl)-26-amino-8-(2-carboxyethyl)-27-hydroxy-23-(hydroxymethyl)-11-isobutyl-5,14-diisopropyl-2,17-dimethyl-4,7,10,13,16,19,22,25-octaoxo-3,6,9,12,15,18,21,24-octaazaheptacosanoic acid
CAS号:114472-81-0
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Pentanedioic acid, mono(2-(dichloroamino)-2-methylpropyl) ester
CAS号:82224-88-2
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3,5-Dichloro-2,4-dimethoxy-6-(trichloromethyl)pyridine
CAS号:108030-77-9
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(S)-6-(((2-amino-3-hydroxy-3-methylbutanoyl)oxy)methyl)-9-methoxyphenazine-1-carboxylic acid
CAS号:173485-80-8
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1-[1-(2-Ethoxyethyl)-3-ethyl-7-[(4-methylpyridin-2-yl)amino]pyrazolo[4,3-d]pyrimidin-5-yl]piperidine-4-carboxylic acid
CAS号:936449-28-4
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phenyl (R)-(1-(3-(3,4-dimethoxyphenyl)-2,6-dimethylimidazo[1,2-b]pyridazin-8-yl)pyrrolidin-3-yl)carbamate
CAS号:2232878-43-0
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2-[[2-(3,4-dichlorophenyl)-1,3-dihydroisoindol-5-yl]amino]pyridine-3-carboxylic acid
CAS号:313533-41-4
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3-[(2S)-2-{[(adamantan-2-yloxy)carbonyl]amino}-2-(1H-indol-3-ylmethyl)propanamido]-4-(4-fluorophenyl)butanoic acid
CAS号:181941-32-2
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(3R)-3-[[(2S)-2-(2-adamantyloxycarbonylamino)-3-(1H-indol-3-yl)-2-methylpropanoyl]amino]-4-phenylbutanoic acid
CAS号:140677-01-6
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(S)-3-((R)-2-(((adamantan-2-yloxy)carbonyl)amino)-3-(1H-indol-3-yl)-2-methylpropanamido)-4-(4-aminophenyl)butanoic acid
CAS号:149027-97-4
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7-(3-(1-aminoethyl)pyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid
CAS号:147208-55-7
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(3S)-3-[[(2R)-2-(2-adamantyloxycarbonylamino)-3-(1H-indol-3-yl)-2-methylpropanoyl]amino]-4-phenylbutanoic acid
CAS号:134557-41-8
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(2S,4S,5S)-N-butyl-6-cyclohexyl-4-hydroxy-2-isopropyl-5-((S)-2-((S)-2-(morpholine-4-sulfonamido)-3-phenylpropanamido)pent-4-enamido)hexanamide
CAS号:150351-30-7
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5-(3-(1H-imidazol-4-yl)-2-(3-(naphthalen-1-yl)-2-(naphthalen-1-ylmethyl)propanamido)propanamido)-6-cyclohexyl-4-hydroxy-2-isobutyl-N-(2-methylbutyl)hexanamide
CAS号:128139-14-0
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1-(4-amino-3-methylbenzyl)-5-(2,2-diphenylacetyl)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridine-6-carboxylic acid
CAS号:114785-12-5
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7-(3-aminopyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid
CAS号:96568-33-1


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